Li-tubes tsa laboratori

Sehlahisoa

Pimobendan 74150-27-9 Metabolism PDE inhibitor

Tlhaloso e Khutšoanyane:

Lebitso la sehlahisoa:Pimobendan
Mantsoe a tšoanang:4,5-Dihydro-6-[2-(4-methoxyphenyl)-1H-benzimidazol-6-yl]-5-methyl-3(2H)-pyridazinone
Nomoro ea CAS:74150-27-9
Boleng:USP43
Foromo ea molek'hule:C19H18N4O2
Boima ba molek'hule:334.37


Lintlha tsa Sehlahisoa

Li-tag tsa Sehlahisoa

Tefo:T/T, L/C
Tšimoloho ea Sehlahisoa:China
Boema-kepe:Beijing/Shanghai/Hangzhou
Odara (MOQ):1g
Lead time:3 matsatsi a ho sebetsa
Bokhoni ba tlhahiso:1kg/khoeli
Boemo ba polokelo:E bolokiloe sebakeng se pholileng, se omileng, mocheso oa kamore.
Lintho tsa sephutheloana:vial, botlolo
Boholo ba sephutheloana:1g/vial, 5/vial, 10g/vial, 50g/botlolo, 500g/botlolo
Lintlha tsa polokeho:UN 2811 6.1/PG 3

Pimobendan

Selelekela

Pimobendan, ke moriana oa bongaka ba liphoofolo.Ke calcium sensitizer le inhibitor e khethiloeng ea phosphodiesterase 3 (PDE3) e nang le liphello tse ntle tsa inotropic le vasodilator.

Pimobendan e sebelisoa ho laola ho hloleha ha pelo ho lintja, hangata ho bakoang ke myxomatous mitral valve disease (eo pele e neng e tsejoa e le endocardiosis), kapa dilated cardiomyopathy.Patlisiso e bonts'itse hore joalo ka monotherapy, pimobendan e eketsa nako ea ho pholoha le ho ntlafatsa boleng ba bophelo ho bakuli ba canine ba nang le ho hloleha ha pelo ho latela lefu la mitral valve ha le bapisoa le benazepril, e leng ACE inhibitor.

Tlhaloso (USP43)

Ntho

Tlhaloso

Ponahalo

Phofo e tšoeu kapa e mosehla hanyenyane, hygroscopic

Mp

Hoo e ka bang 242 ℃

Solubility

Ha e khone ho qhibiliha ka metsing, e qhibiliha ka bolokolohi ho dimethylformamide, e qhibiliha hanyenyane ho acetone le methanil.

Boitsebiso

Infrared absorption spectrophotometry, Papiso ea pimobendan CRS.

Nako ea ho boloka tlhōrō e kholo ea tharollo ea Sample e lumellana le ea Standard stock solution, joalokaha e fumanoe tekong ea Organic Impurities.

Litšepe tse boima

≤10ppm

Granularity

P90 ≤ 25μ m

Boholo ba likaroloana

20-80 mesh

Li-solvents tse setseng

≤ 500ppm

Metsi

≤ 1.0%

Tlhahlobo

98.0%~102.0%

Molora o nang le sulphated

≤ 0.10%

Lintho tse amanang le tsona (HPLC)

litšila A

≤ 0.10%

litšila B

≤ 0.10%

Tšilafalo efe kapa efe

≤ 0.10%

Ho se hloeke ho feletseng

≤ 0.20%


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